Histamine Receptor Inhibitor

Histamine Receptor Inhibitors (47):

Cat. No.	Product Name	Effect	Purity

HY-N0054

Osthole	Inhibitor	99.95%
Osthole (Osthol) is a natural antihistamine alternative. Osthole may be a potential inhibitor of histamine H₁ receptor activity. Osthole also suppresses the secretion of HBV in cells.

HY-14270

Lodoxamide	Inhibitor	98.07%
Lodoxamide (U-42585E free acid) is an antiallergic compound acting as a mast-cell stabilizer for the treatment of asthma and allergic conjunctivitis.

HY-12199

Pitolisant	Inhibitor
Pitolisant is a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (K_i=0.16 nM).

HY-B1062

Dexchlorpheniramine maleate	Inhibitor	≥98.0%
Dexchlorpheniramine maleate is an antihistamine, with anticholinergic properties, used to treat allergic conditions.

HY-B0170A

Azatadine dimaleate	Inhibitor	99.85%
Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.

HY-B0426A

Olopatadine hydrochloride	Inhibitor	99.71%
Olopatadine hydrochloride (ALO4943A) is a histamine blocker used to treat allergic conjunctivitis.

HY-B1090

Cinnarizine	Inhibitor	99.63%
Cinnarizine is an antihistamine and a calcium channel blocker, promote cerebral blood flow, used to treat cerebral apoplexy, post-trauma cerebral symptoms, and cerebral arteriosclerosis.

HY-B0801S

Fexofenadine-d₆	Inhibitor	99.28%
Fexofenadine-d₆ is deuterium labeled Fexofenadine, which is an antihistamine pharmaceutical agent.

HY-B1510

Acrivastine	Inhibitor	99.59%
Acrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis.

HY-B1895

Levodropropizine	Inhibitor	99.71%
Levodropropizine (DF-526) is an orally active histamine receptor inhibitor, Levodropropizine is an effective and very well tolerated peripheral antitussive agent.

HY-16289

Lodoxamide tromethamine	Inhibitor	99.85%
Lodoxamide tromethamine (U-42585E) is a medication for the treatment of prophylaxis of mast cell-mediated allergic disease.

HY-B1067

Antazoline hydrochloride	Inhibitor	99.70%
Antazoline hydrochloride is a 1st generation antihistamine with also anticholinergic properties used to relieve nasal congestion and in eye drops.

HY-B0527AS

Amitriptyline-d₆ hydrochloride	Inhibitor	99.65%
Amitriptyline-d₆ (hydrochloride) is the deuterium labeled Amitriptyline hydrochloride. Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with Kis of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a Ki of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic, muscarinic, histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity[1][2][3].

HY-135096

Amitriptyline-d3 hydrochloride	Inhibitor	99.46%
Amitriptyline-d3 hydrochloride is the deuterium labeled Amitriptyline (hydrochloride). Amitriptyline hydrochloride is an inhibitor of serotonin reuptake transporter (SERT) and noradrenaline reuptake transporter (NET), with K_is of 3.45 nM and 13.3 nM for human SERT and NET, respectively. Amitriptyline hydrochloride also weakly binds to dopamine reuptake transporter (DAT) with a K_i of 2.58 μM. Amitriptyline hydrochloride also inhibits adrenergic, muscarinic, histamine and 5-HT receptors. Amitriptyline hydrochloride is a TrkA and TrkB receptors agonist with potent neurotrophic activity. Amitriptyline hydrochloride has antidepressant activity.

HY-B0530

Azacyclonol	Inhibitor	99.99%
Azacyclonol (γ-pipradol), a metabolite of Terfenadine, is a central depressant agent. Azacyclonol is a ganglion-blocking agent. Azacyclonol can be used to diminish psychoses-induced hallucinations.

HY-109544

Repirinast	Inhibitor
Repirinast (MY-5116) is an orally active anti-allergic agent. Repirinast inhibits histamine release. Repirinast can be used in the research of bronchial asthma.

HY-B1607

Chlorphenoxamine	Inhibitor
Chlorphenoxamine is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.

HY-B0188

Mianserin	Inhibitor
Mianserin is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.

HY-B1395A

Mecamylamine	Inhibitor
Mecamylamine is an orally active, nonselective, noncompetitive nAChR antagonist. Mecamylamine is also a ganglionic blocker. Mecamylamine can across the blood-brain barrier. Mecamylamine can be used in the research of neuropsychiatric disorders, hypertension, antidepressant area.

HY-139519S

N-Desmethyl diphenhydramine-d₃ hydrochloride	Inhibitor
N-Desmethyl diphenhydramine-d₃ (hydrochloride) is the deuterium labeled N-Desmethyl diphenhydramine hydrochloride[1].

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